Published 2013
Table of Contents:
“…Assay Considerations for Compound Library
Screening.4.1 Defining Inhibition Signal Robustness, and Hit Criteria.4.
2 Measuring Initial Velocity.4.
2.1 End-Point and Kinetic Readouts.4.
2.
2 Effects of Enzyme Concentration.4.3 Balanced Assay Conditions.4.3.1 Balancing Conditions for Multisubstrate Reactions.4.4 Order of Reagent Addition.4.5 Use of Natural Substrates and Enzymes.4.6 Coupled Enzyme Assays.4.7 Hit Validation and Progression.4.8 Summary.References.5. …”
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